Popular99%+ Purity

AICAR

AMPK activator / exercise mimetic

Available Forms
Lyophilized Powder
Total$1,000.00

100 unit minimum per SKU • Wholesale pricing

Why Choose Scientific Aminos?

Certificate of Analysis

Every batch tested with COA provided

99%+ Purity

HPLC verified purity standards

US Manufacturing

cGMP compliant facilities

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Research Areas
AMPK SignalingExercise PhysiologyMetabolic ResearchEndurance Studies

AMPK activator for metabolic and exercise research. AICAR (5-Aminoimidazole-4-carboxamide ribonucleotide) is a cell-permeable AMPK activator that mimics exercise-induced metabolic changes.

AICAR Research Compound

Research Use Only

This product is intended for laboratory research purposes only. It is not intended for human or veterinary use, food, cosmetic, household, or agricultural applications. Not for human consumption.

Overview

AICAR (5-Aminoimidazole-4-carboxamide ribonucleotide, also known as Acadesine) is a cell-permeable nucleoside analog that activates AMP-activated protein kinase (AMPK). Often called an "exercise mimetic," AICAR triggers many of the same metabolic adaptations as endurance exercise.

Mechanism of Action

AICAR activates AMPK through:

  • Conversion to ZMP (AICAR monophosphate)
  • Direct AMPK activation (mimics AMP)
  • Enhanced glucose uptake
  • Increased fatty acid oxidation
  • Mitochondrial biogenesis stimulation

Exercise Mimetic Effects

EffectExerciseAICAR
AMPK Activation++
Glucose Uptake++
Fat Oxidation++
Mitochondrial Biogenesis++
PGC-1alpha Activation++

Research Applications

  • AMPK pathway studies
  • Exercise physiology research
  • Metabolic adaptation mechanisms
  • Endurance capacity studies

Handling & Storage

  • Store lyophilized powder at -20C
  • Protect from light and moisture
  • Reconstitute with sterile water
  • Reconstituted solution stable at 2-8C for up to 1 week

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